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GluK1 antagonists from 6-(tetrazolyl)phenyl decahydroisoquinoline derivatives: In vitro profile and in vivo analgesic efficacy

José Antonio Martínez-Pérez, Smriti Iyengar, Harlan E. Shannon, David Bleakman, Andrew Alt, David K. Clawson, Brian M. Arnold, Michael G. Bell, Thomas J. Bleisch, Ana M. Castaño‐León,

Bioorganic & Medicinal Chemistry Letters · 2013 · 10 citations · 15 references

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15

Crystal Structures of the GluR5 and GluR6 Ligand Binding Cores: Molecular Mechanisms Underlying Kainate Receptor Selectivity

Mark L. Mayer · Neuron · 2005 · 260 citations · Full text

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Total synthesis of 1233A

Peter M. Wovkulich, K. Shankaran, Milan R. Uskoković · The Journal of Organic Chemistry · 1993 · 191 citations

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LY293558, a Novel AMPA/GluR5 Antagonist, is Efficacious and Well-Tolerated in Acute Migraine

CN Sang, NM Ramadan, RG Wallihan et al. · Cephalalgia · 2004 · 173 citations

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Kainate GluR5 receptor subtype mediates the nociceptive response to formalin in the rat

Rosa Maria A. Simmons, Dominic L. Li, Ken H. Hoo et al. · Neuropharmacology · 1998 · 172 citations

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AMPA/Kainate Antagonist LY293558 Reduces Capsaicin-evoked Hyperalgesia but Not Pain in Normal Skin in Humans 

Christine N. Sang, Meredith P. Hostetter, Richard H. Gracely et al. · Anesthesiology · 1998 · 130 citations · Full text

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