Thomas J. Bleisch

2-Substituted (2<i>SR</i>)-2-Amino-2-((1<i>SR</i>,2<i>SR</i>)-2-carboxycycloprop-1-yl)glycines as Potent and Selective Antagonists of Group II Metabotropic Glutamate Receptors. 2. Effects of Aromatic Substitution, Pharmacological Characterization, and Bioavailability

Paul L. Ornstein, Thomas J. Bleisch, M. Brian Arnold et al. · Journal of Medicinal Chemistry · 1998 · 100 citations · Full text

Pharmacological Characterization, Synaptic Transmission, Pharmacotherapy +19

Biarylpropylsulfonamides as Novel, Potent Potentiators of 2-Amino-3- (5-methyl-3-hydroxyisoxazol-4-yl)- propanoic Acid (AMPA) Receptors

Paul L. Ornstein, Dennis M. Zimmerman, M. Brian Arnold et al. · Journal of Medicinal Chemistry · 2000 · 75 citations · Full text

Pharmaceutical Science, Potent Potentiators, Altmetric Attention Score +17

2-Substituted (2<i>SR</i>)-2-Amino-2-((1<i>SR</i>,2<i>SR</i>)-2-carboxycycloprop-1-yl)glycines as Potent and Selective Antagonists of Group II Metabotropic Glutamate Receptors. 1. Effects of Alkyl, Arylalkyl, and Diarylalkyl Substitution

Paul L. Ornstein, Thomas J. Bleisch, M. Brian Arnold et al. · Journal of Medicinal Chemistry · 1998 · 72 citations · Full text

Ethyl (3<i>S</i>,4a<i>R</i>,6<i>S</i>,8a<i>R</i>)-6-(4-Ethoxycar- bonylimidazol-1-ylmethyl)decahydroiso- quinoline-3-carboxylic Ester:  A Prodrug of a GluR5 Kainate Receptor Antagonist Active in Two Animal Models of Acute Migraine

Sandra Filla, Mark A. Winter, Kirk W. Johnson et al. · Journal of Medicinal Chemistry · 2002 · 51 citations · Full text

Diethyl Ester, Pharmacotherapy, Experimental Pharmacology +22

Novel 3-Aryl Indoles as Progesterone Receptor Antagonists for Uterine Fibroids

Timothy I. Richardson, Christian A. Clarke, Kuo‐Long Yu et al. · ACS Medicinal Chemistry Letters · 2010 · 50 citations · Full text

Medicinal Chemistry, Hormonal Contraceptive, Uterine Fibroids +15