Mark A. Winter

Molecular determinants of tissue selectivity in estrogen receptor modulators

Timothy A. Grese, James P. Sluka, Henry U. Bryant et al. · Proceedings of the National Academy of Sciences · 1997 · 242 citations · Full text

Estrogen Receptor, Gynecology, Raloxifene Analogs +16

Essential features of the P-glycoprotein pharmacophore as defined by a series of reserpine analogs that modulate multidrug resistance.

Homer L. Pearce, Ahmad R. Safa, Nicholas J. Bach et al. · Proceedings of the National Academy of Sciences · 1989 · 234 citations · Full text

Drug Target, P-glycoprotein Pharmacophore, Pharmacotherapy +18

Application of Three-Dimensional Quantitative Structure-Activity Relationships of P-Glycoprotein Inhibitors and Substrates

Sean Ekins, Richard B. Kim, Brenda F. Leake et al. · Molecular Pharmacology · 2002 · 185 citations

Structure−Activity Relationships of Selective Estrogen Receptor Modulators:  Modifications to the 2-Arylbenzothiophene Core of Raloxifene

Timothy A. Grese, Stephen Cho, Don R. Finley et al. · Journal of Medicinal Chemistry · 1997 · 175 citations · Full text

Gynecology, Raloxifene Analogs, Pharmacotherapy +23

Three-Dimensional Quantitative Structure-Activity Relationships of Inhibitors of P-Glycoprotein

Sean Ekins, Richard B. Kim, Brenda F. Leake et al. · Molecular Pharmacology · 2002 · 166 citations · Full text