Synthesis of enantiopure azetidine 2-carboxylic acids and their incorporation into peptides

Peptidomimetics for Receptor Ligands—Discovery, Development, and Medical Perspectives

Athanassios Giannis, Thomas Kolter · Angewandte Chemie International Edition in English · 1993 · 778 citations

Peptide Engineering, Pharmacotherapy, Receptor Ligands—discovery +17

Design and synthesis of conformationally constrained amino acids as versatile scaffolds and peptide mimetics

Stephen Hanessian, Grant McNaughton‐Smith, Henry‐Georges Lombart et al. · Tetrahedron · 1997 · 629 citations

Peptide Mimetics, Amino Acids, Biochemistry +12

Cyclopropane amino acids

Charles H. Stammer · Tetrahedron · 1990 · 307 citations

Cyclopropane Amino Acids, Heterocyclic, Biochemistry +1

Towards control of χ-space: Conformationally constrained analogues of Phe, Tyr, Trp and His

Susan E. Gibson, Nathalie Guillo, Matthew J. Tozer · Tetrahedron · 1999 · 219 citations

Quantum Field Theory, Conformational Study, Towards Control +2

Cyclic amino acid derivatives

Mark J. Kurth · Tetrahedron · 2002 · 169 citations

Derivative (Chemistry), Bioorganic Chemistry, Biochemistry +4