Henry‐Georges Lombart

Design and synthesis of conformationally constrained amino acids as versatile scaffolds and peptide mimetics

Stephen Hanessian, Grant McNaughton‐Smith, Henry‐Georges Lombart et al. · Tetrahedron · 1997 · 629 citations

Peptide Mimetics, Amino Acids, Biochemistry +12

Rigid Dipeptide Mimetics:  Efficient Synthesis of Enantiopure Indolizidinone Amino Acids

Henry‐Georges Lombart, William D. Lubell · The Journal of Organic Chemistry · 1996 · 66 citations

Combinatorial Chemistry, Rigid Dipeptide Mimetics, Inexpensive Glutamic Acid +16

Total Synthesis of Elaiolide Using a Copper(I)-Promoted Stille Cyclodimerization Reaction

Ian Paterson, Henry‐Georges Lombart, Charlotte Allerton · Organic Letters · 1999 · 64 citations

Bioorganic Chemistry, Engineering, Organic Chemistry +16

Synthesis of Enantiopure .alpha.,.omega.-Diamino Dicarboxylates and Azabicycloalkane Amino Acids by Claisen Condensation of .alpha.-[N-(Phenylfluorenyl)amino] Dicarboxylates

Henry‐Georges Lombart, William D. Lubell · The Journal of Organic Chemistry · 1994 · 62 citations

Combinatorial Chemistry, Bioorganic Chemistry, Engineering +18

Identification of potent and selective TACE inhibitors via the S1 pocket

Jeffrey S. Condon, Diane Joseph‐McCarthy, Jeremy I. Levin et al. · Bioorganic & Medicinal Chemistry Letters · 2006 · 39 citations · Full text

Selective Tace Inhibitors, Medicinal Chemistry, Drug Target +11