Concepedia

Synthesis, inhibition and binding of simple non-nitrogen inhibitors of monoamine transporters

Mikkel Due Petersen, Søren V. Boye, Erik Nguyen Nielsen, Jeanette Willumsen, Steffen Sinning, Ove Wiborg, Mikael Bols

Bioorganic & Medicinal Chemistry · 2007 · 22 citations · 21 references

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21

Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

Yung-Chi Cheng, William H. Prusoff · Biochemical Pharmacology · 1973 · 12.9K citations

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Compounds Affecting the Central Nervous System. 4. 3.beta.-Phenyltropane-2-carboxylic Esters and Analogs

Robert B. Clarke, Sol J. Daum, A. J. GAMBINO et al. · Journal of Medicinal Chemistry · 1973 · 217 citations

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Microwave-Assisted Synthesis of Pinacol Boronates from Aryl Chlorides Catalyzed by a Palladium/Imidazolium Salt System

Alois Fürstner, Günter Seidel · Organic Letters · 2002 · 158 citations

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Synthesis, ligand binding, QSAR, and CoMFA study of 3.beta.-(p-substituted phenyl)tropane-2.beta.-carboxylic acid methyl esters

F. Ivy Carroll, Yigong Gao, M. Abdur Rahman et al. · Journal of Medicinal Chemistry · 1991 · 146 citations · Full text

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Monoamine transporter gene structure and polymorphisms in relation to psychiatric and other complex disorders

Maureen K. Hahn, Randy Blakely · The Pharmacogenomics Journal · 2002 · 140 citations

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