Efficient preparation of an N-aryl β-amino acid via asymmetric hydrogenation and direct asymmetric reductive amination en route to Ezetimibe

Guuske F. Busscher, Laurent Lefort, Jozef G.O. Cremers, Marco Mottinelli, Roel W. Wiertz, Ben de Lange, Yutaka Okamura, Yukinori Yusa, Kazuhiko Matsumura, Hideo Shimizu,

Tetrahedron Asymmetry · 2010 · 41 citations · 34 references

DOIFull text

Open access

Concepts

References

34