Biological activities of cyclic enkephalin pseudopeptides containing thioamides as amide bond replacements

EFFECT OF MORPHINE ON ADRENERGIC TRANSMISSION IN THE MOUSE VAS DEFERENS. ASSESSMENT OF AGONIST AND ANTAGONIST POTENCIES OF NARCOTIC ANALGESICS

Joel W. Hughes, H. W. Kosterlitz, Frances M. Leslie · British Journal of Pharmacology · 1975 · 405 citations · Full text

Medicine, Pharmacology, Neuropharmacology +11

The effects of adrenaline, noradrenaline and isoprenaline on inhibitory α‐ and β‐adrenoceptors in the longitudinal muscle of the guinea‐pig ileum

H. W. Kosterlitz, R. J. LYDON, A Watt · British Journal of Pharmacology · 1970 · 362 citations · Full text

Medicine, Pharmacology, Physiology +12

Molecular mechanism of opioid receptor selection

R. Schwyzer · Biochemistry · 1986 · 258 citations

Medicine, Pharmacology, Molecular Pharmacology +6

Synthesis and pharmacological characterization in vitro of cyclic enkephalin analogs: effect of conformational constraints on opiate receptor selectivity

John DiMaio, Thi M.‐D. Nguyen, Carole Lemieux et al. · Journal of Medicinal Chemistry · 1982 · 200 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +11

Dermorphin analogs carrying an increased positive net charge in their "message" domain display extremely high .mu.-opioid receptor selectivity

Peter W. Schiller, Nguyen Thi Mai Dung, Nga N. Chung et al. · Journal of Medicinal Chemistry · 1989 · 169 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +15