Carole Lemieux

Synthesis and pharmacological characterization in vitro of cyclic enkephalin analogs: effect of conformational constraints on opiate receptor selectivity

John DiMaio, Thi M.‐D. Nguyen, Carole Lemieux et al. · Journal of Medicinal Chemistry · 1982 · 200 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +11

The Opioid μ Agonist/δ Antagonist DIPP-NH₂[Ψ] Produces a Potent Analgesic Effect, No Physical Dependence, and Less Tolerance than Morphine in Rats

Peter W. Schiller, Marian E. Fundytus, Lisa Merovitz et al. · Journal of Medicinal Chemistry · 1999 · 188 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +17

Dermorphin analogs carrying an increased positive net charge in their "message" domain display extremely high .mu.-opioid receptor selectivity

Peter W. Schiller, Nguyen Thi Mai Dung, Nga N. Chung et al. · Journal of Medicinal Chemistry · 1989 · 169 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +15

Synthesis and in vitro opioid activity profiles of DALDA analogues

Peter W. Schiller, Thi M.‐D. Nguyen, Irena Berezowska et al. · European Journal of Medicinal Chemistry · 2000 · 161 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +12

TIPP[.psi.]: a highly potent and stable pseudopeptide .delta. opioid receptor antagonist with extraordinary .delta. selectivity

Peter W. Schiller, Grazyna Weltrowska, Thi M.‐D. Nguyen et al. · Journal of Medicinal Chemistry · 1993 · 147 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +16