Quinine as chiral discriminator for determination of enantiomeric excess of diethyl 1,2-dihydroxyalkanephosphonates

The osmium-catalyzed asymmetric dihydroxylation: a new ligand class and a process improvement

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Natural Sciences, Biochemistry, Chemistry +7

New hybrid transition state analog inhibitors of HIV protease with peripheric C2-symmetry

Bernd Stowasser, Karl‐Heinz Budt, Jianqi Li et al. · Tetrahedron Letters · 1992 · 407 citations

Life Sciences, Medicinal Chemistry, Molecular Biology +13

Preparation of peptidic α-hydroxy phosphonates a new class of transition state analog renin inhibitors

Dinesh V. Patel, Katherine Rielly-Gauvin, Denis E. Ryono · Tetrahedron Letters · 1990 · 237 citations

Pharmacy, Medicinal Chemistry, Pharmacology +12

.alpha.-Hydroxy Phosphinyl-Based Inhibitors of Human Renin

Dinesh V. Patel, Katherine Rielly-Gauvin, Denis E. Ryono et al. · Journal of Medicinal Chemistry · 1995 · 193 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +15

The Catalytic Asymmetric Aminohydroxylation of Unsaturated Phosphonates

Allen A. Thomas, K. Barry Sharpless · The Journal of Organic Chemistry · 1999 · 123 citations

Pharmacy, Biochemistry, Chemistry +6