Concepedia

2-Phenyl-4-piperazinylbenzimidazoles: Orally active inhibitors of the gonadotropin releasing hormone (GnRH) receptor

Jeffrey C. Pelletier, Murty Chengalvala, Josh Cottom, Irene Feingold, Lloyd Garrick, Daniel J. Green, Diane B. Hauze, Christine Huselton, James W. Jetter, Wenling Kao

Bioorganic & Medicinal Chemistry · 2008 · 29 citations · 17 references

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17

Experimental and computational approaches to estimate solubility and permeability in drug discovery and development settings

Christopher A. Lipinski, Franco Lombardo, Beryl W. Dominy et al. · Advanced Drug Delivery Reviews · 1997 · 11.2K citations

, , +16

Molecular Properties That Influence the Oral Bioavailability of Drug Candidates

Daniel F. Veber, Stephen R. Johnson, Hung‐Yuan Cheng et al. · Journal of Medicinal Chemistry · 2002 · 8.1K citations

, , +15

Structure of the porcine LH- and FSH-releasing hormone. I. The proposed amino acid sequence

H. Matsuo, Akira Arimura, Andrew V. Schally · Biochemical and Biophysical Research Communications · 1971 · 1.1K citations

, , +16

Structure of the porcine LH- and FSH-releasing hormone. I. The proposed amino acid sequence

American Journal of Obstetrics and Gynecology · 1976 · 1K citations

, , +16

Gonadotropin-Releasing Hormone: One Polypeptide Regulates Secretion of Luteinizing and Follicle-Stimulating Hormones

Andrew V. Schally, Akira Arimura, Abba J. Kastin et al. · Science · 1971 · 759 citations

, , +15