Stereodivergent synthesis of β-amino-α-hydroxyphosphonic acid derivatives by lewis acid mediated stereosclective hydrophosphonylation of α-amino aldehydes

New hybrid transition state analog inhibitors of HIV protease with peripheric C2-symmetry

Bernd Stowasser, Karl‐Heinz Budt, Jianqi Li et al. · Tetrahedron Letters · 1992 · 407 citations

Life Sciences, Medicinal Chemistry, Molecular Biology +13

Preparation of peptidic α-hydroxy phosphonates a new class of transition state analog renin inhibitors

Dinesh V. Patel, Katherine Rielly-Gauvin, Denis E. Ryono · Tetrahedron Letters · 1990 · 237 citations

Pharmacy, Medicinal Chemistry, Pharmacology +12

New silicon-phosphorus reagents in organic synthesis. Carbonyl and conjugate addition reactions of silicon phosphite esters and related systems

David A. Evans, K. M. HURST, James M. Takacs · Journal of the American Chemical Society · 1978 · 140 citations

Natural Sciences, Chemistry, Inorganic Chemistry +6

Aluminoxy acetals from .alpha.-amino esters: chirality transfer via sequential addition of hydride and C-nucleophiles. 2-Amino alcohols and sphingosines

Robin Polt, Matt A. Peterson · The Journal of Organic Chemistry · 1992 · 110 citations

Natural Sciences, Biochemistry, Chemistry +10

Peptidic α-hydroxy phosphinyls C-terminal modification methodology

Dinesh V. Patel, Katherine Rielly-Gauvin, Denis E. Ryono · Tetrahedron Letters · 1990 · 102 citations

Natural Sciences, Biochemistry, Bioorthogonal Chemistry +2