1-(2-Nitrophenyl)thiosemicarbazides: A Novel Class of Potent, Orally Active Non-Peptide Antagonist for the Bradykinin B₂ Receptor

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ADVERTISEMENT RETURN TO ISSUEPREVLetterNEXT1-(2-Nitrophenyl)thiosemicarbazides: A Novel Class of Potent, Orally Active Non-Peptide Antagonist for the Bradykinin B2 ReceptorEdward K. Dziadulewicz, Timothy J. Ritchie, Allan Hallett, Christopher R. Snell, Soo Y. Ko, Roger Wrigglesworth, Glyn A. Hughes, Andrew R. Dunstan, Graham C. Bloomfield, Gillian S. Drake, Michael C. Brown, Wai Lee, Gillian M. Burgess, Clare Davis, Mohammed Yaqoob, Martin N. Perkins, Elizabeth A. Campbell, Andrew J. Davis, and Humphrey P. RangView Author Information Departments of Medicinal Chemistry, Biology, and Pharmacology, Novartis Institute for Medical Sciences, 5 Gower Place, London WC1E 6BN, England Cite this: J. Med. Chem. 2000, 43, 5, 769–771Publication Date (Web):February 12, 2000Publication History Received3 September 1999Published online12 February 2000Published inissue 1 March 2000https://pubs.acs.org/doi/10.1021/jm991155ohttps://doi.org/10.1021/jm991155orapid-communicationACS PublicationsCopyright © 2000 American Chemical SocietyRequest reuse permissionsArticle Views602Altmetric-Citations26LEARN ABOUT THESE METRICSArticle Views are the COUNTER-compliant sum of full text article downloads since November 2008 (both PDF and HTML) across all institutions and individuals. These metrics are regularly updated to reflect usage leading up to the last few days.Citations are the number of other articles citing this article, calculated by Crossref and updated daily. Find more information about Crossref citation counts.The Altmetric Attention Score is a quantitative measure of the attention that a research article has received online. Clicking on the donut icon will load a page at altmetric.com with additional details about the score and the social media presence for the given article. Find more information on the Altmetric Attention Score and how the score is calculated. Share Add toView InAdd Full Text with ReferenceAdd Description ExportRISCitationCitation and abstractCitation and referencesMore Options Share onFacebookTwitterWechatLinked InRedditEmail Other access optionsGet e-Alertsclose SUBJECTS:Antagonists,Molecules,Peptides and proteins,Receptors,Rodent models Get e-Alerts