Edward K. Dziadulewicz

Synthesis of Nonproteinogenic (<i>R</i>)‐ or (<i>S</i>)‐Amino Acids Analogues of Phenylalanine, Isotopically Labelled and Cyclic Amino Acids from <i>tert</i>‐Butyl 2‐(<i>tert</i>‐Butyl)‐3‐methyl‐4‐oxo‐1‐imidazolidinecarboxylate (Boc‐BMI)

Dieter Seebàch, Edward K. Dziadulewicz, Linda Behrendt et al. · Liebigs Annalen der Chemie · 1989 · 119 citations

Pharmacy, Biochemistry, Medicinal Chemistry +10

Bradyzide, a potent non‐peptide B₂ bradykinin receptor antagonist with long‐lasting oral activity in animal models of inflammatory hyperalgesia

Gillian M. Burgess, Martin Perkins, H P Rang et al. · British Journal of Pharmacology · 2000 · 104 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +11

Naphthalen-1-yl-(4-pentyloxynaphthalen-1-yl)methanone:  A Potent, Orally Bioavailable Human CB₁/CB₂Dual Agonist with Antihyperalgesic Properties and Restricted Central Nervous System Penetration

Edward K. Dziadulewicz, Stuart Bevan, Christopher T. Brain et al. · Journal of Medicinal Chemistry · 2007 · 96 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +16

Identification and Biological Characterization of 6-Aryl-7-isopropylquinazolinones as Novel TRPV1 Antagonists that Are Effective in Models of Chronic Pain

Andrew J. Culshaw, Stuart Bevan, Martin Lau Christiansen et al. · Journal of Medicinal Chemistry · 2005 · 60 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +17

The design of non-peptide human bradykinin B2 receptor antagonists employing the benzodiazepine peptidomimetic scaffold

Edward K. Dziadulewicz, Michael C. Brown, Andrew R. Dunstan et al. · Bioorganic & Medicinal Chemistry Letters · 1999 · 57 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +12