Concepedia
Bioorganic & Medicinal Chemistry Letters · 2001 · 22 citations · 2 references
Open access
Life SciencesMedicinal ChemistryPharmacologyDrug DiscoveryEnzymologySynthetic Medicinal ChemistryEnzyme ActivatorsEnzyme InhibitionLigand BindingEnzyme Inhibitor SynthesisMatrix Metalloproteinase Inhibitors
2
Discovery of Potent Nonpeptide Inhibitors of Stromelysin Using SAR by NMR
Philip J. Hajduk, George S. Sheppard, David G. Nettesheim et al. · Journal of the American Chemical Society · 1997 · 317 citations
Pharmacy, Medicinal Chemistry, Pharmacology +13
Design, Synthesis, and Biological Evaluation of Matrix Metalloproteinase Inhibitors Derived from a Modified Proline Scaffold
Menyan Cheng, Biswanath De, Neil G. Almstead et al. · Journal of Medicinal Chemistry · 1999 · 51 citations · Full text
Pharmacy, Chemistry, Medicinal Chemistry +17