New insights in endogenous modulation of ligand-gated ion channels: Histamine is an inverse agonist at strychnine sensitive glycine receptors

Auto-inhibition of brain histamine release mediated by a novel class (H3) of histamine receptor

Jean‐Michel Arrang, M. Garbarg, Jean‐Charles Schwartz · Nature · 1983 · 1.6K citations

Life Sciences, Neuroscience, Pharmacology +14

The β Subunit Determines the Ligand Binding Properties of Synaptic Glycine Receptors

Joanna Grudzinska, Rudolf Schemm, Svenja Haeger et al. · Neuron · 2005 · 357 citations · Full text

Life Sciences, Neurobiology, Neuroscience +16

The atypical M2 segment of the beta subunit confers picrotoxinin resistance to inhibitory glycine receptor channels.

I. Pribilla, T. Takagi, Dieter Langosch et al. · The EMBO Journal · 1992 · 317 citations · Full text

Medicine, Molecular Biology, Pharmacology +7

Analysis of the Set of GABAA Receptor Genes in the Human Genome

Joseph Simon, Hironobu Wakimoto, Norihisa Fujita et al. · Journal of Biological Chemistry · 2004 · 255 citations · Full text

Life Sciences, Genetics, Neuroscience +8

Residues within transmembrane segment M2 determine chloride conductance of glycine receptor homo‐ and hetero‐oligomers.

Joachim Bormann, N. Rundström, Heinrich Betz et al. · The EMBO Journal · 1993 · 247 citations

Natural Sciences, Biochemistry, Biophysics +11