Concepedia

Discovery of ‘molecular switches’ within a GIRK activator scaffold that afford selective GIRK inhibitors

Wandong Wen, Wenjun Wu, Ian M. Romaine, Kristian Kaufmann, Yu Du, Gary A. Sulikowski, C. David Weaver, Craig W. Lindsley

Bioorganic & Medicinal Chemistry Letters · 2013 · 27 citations · 13 references

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References

13

The G-protein-gated atrial K+ channel IKAch is a heteromultimer of two inwardly rectifying K+-channel proteins

Grigory Krapivinsky, Eric A. Gordon, Kevin Wickman et al. · Nature · 1995 · 845 citations

, , +14

Primary structure and functional expression of a rat G-protein-coupled muscarinic potassium channel

Yoshihiro Kubo, Eitan Reuveny, Paul A. Slesinger et al. · Nature · 1993 · 600 citations

, , +16

IRK(1–3) and GIRK(1–4) Inwardly Rectifying K<sup>+</sup>Channel mRNAs Are Differentially Expressed in the Adult Rat Brain

Christine Karschin, Walter Stühmer, Andreas Karschin · Journal of Neuroscience · 1996 · 451 citations · Full text

, , +14

Cloning provides evidence for a family of inward rectifier and G‐protein coupled K<sup>+</sup> channels in the brain

Florian Lesage, Fabrice Duprat, Michel Fink et al. · FEBS Letters · 1994 · 281 citations

, , +16

Ethanol opens G-protein-activated inwardly rectifying K+ channels

Toru Kobayashi, Kazutaka Ikeda, Hiroshi Kojima et al. · Nature Neuroscience · 1999 · 258 citations

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