5-Vinyl-3-pyridinecarbonitrile inhibitors of PKCθ: Optimization of enzymatic and functional activity

L. Nathan Tumey, Niala Bhagirath, Agnes Brennan, Natasja Brooijmans, Julie Lee, Xiaoke Yang, Diane H. Boschelli

Bioorganic & Medicinal Chemistry · 2009 · 26 citations · 30 references

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