Characterization of human serotonin 1D and 1B receptors using [ 3H]-GR-125743, a novel radiolabelled serotonin 5HT1D/1B receptor antagonist

References

Page 1

	Year	Citations
A Rapid and Sensitive Method for the Quantitation of Microgram Quantities of Protein Utilizing the Principle of Protein-Dye Binding Mark A. Bradford Analytical Biochemistry Protein ChemistryBiochemistryProtein FoldingMicrogram QuantitiesBioanalysis	1976	225.3K
A ternary complex model explains the agonist-specific binding properties of the adenylate cyclase-coupled beta-adrenergic receptor. A. De Léan, Jeffrey M. Stadel, Robert J. Lefkowitz Journal of Biological Chemistry Agonist-specific Binding PropertiesExperimental PharmacologyTernary Complex HrxMolecular PharmacologyTernary Complex Model	1980	1.6K
Characterization of a novel 3H-5-hydroxytryptamine binding site subtype in bovine brain membranes RE Heuring, SJ Peroutka Journal of Neuroscience	1987	404
GR43175, a selective agonist for the 5‐HT<sub>1</sub>‐like receptor in dog isolated saphenous vein P.P.A. Humphrey, W. Feniuk, M.J. Perren, British Journal of Pharmacology Animal PhysiologyMolecular PharmacologySaphenous VeinSignal TransductionMolecular Physiology	1988	300
Human serotonin 1D receptor is encoded by a subfamily of two distinct genes: 5-HT1D alpha and 5-HT1D beta. Richard L. Weinshank, J M Zgombick, M Macchi, Proceedings of the National Academy of Sciences GeneticsNeurotransmitterDistinct GenesMolecular Pharmacology5-Ht1d Alpha	1992	293
Characterization of the 5-HTIB recognition site in rat brain: Binding studies with (−)[125I]Iodocyanopindolol Daniël Hoyer, G. Engel, Hans O. Kalkman European Journal of Pharmacology Neuroimaging BiomarkersNeurophysiologyCellular NeuroscienceNeuropharmacologyBrain Science	1985	281
Molecular cloning and characterization of a rat brain cDNA encoding a 5-hydroxytryptamine1B receptor. Mark M. Voigt, D. J. Laurie, P. H. Seeburg, The EMBO Journal Molecular NeuroscienceMedicineRat Brain CdnaNeurotransmitterNeuropharmacology	1991	217
POSSIBLE BENEFIT OF GR43175, A NOVEL 5-HT1-LIKE RECEPTOR AGONIST, FOR THE ACUTE TREATMENT OF SEVERE MIGRAINE Jochen Brand, V.L. Perrin The Lancet Functional SelectivityMedicineNeuropharmacologyNeurologyNeuroscience	1988	186
5-HT1D as well as 5-HT1A autoreceptors modulate 5-HT release in the guinea-pig dorsal raphénucleus Sarah J. Starkey, M. Skingle Neuropharmacology Animal Physiology5-Ht ReleaseNeurophysiology5-Ht1a AutoreceptorsPhysiology	1994	156
Molecular cloning and functional characterization of a human 5-HT1B serotonin receptor: A homologue of the rat 5-HT1B receptor with 5-HT1D-like pharmacological specificity Mark W. Hamblin, Mark A. Metcalf, Robert W. McGuffin, Biochemical and Biophysical Research Communications Molecular PharmacologyFunctional SelectivityMedicineNeurotransmitterRat 5-Ht1b Receptor	1992	117

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