New insight into active muscarinic receptors with the novel radioagonist [3H]iperoxo

Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

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Cent Inhibition, Inhibitory Activity, Biochemistry +8

Crystal structure of the β2 adrenergic receptor–Gs protein complex

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Molecular Pharmacology, Crystal Structure, Biochemistry +6

The G-Protein-Coupled Receptors in the Human Genome Form Five Main Families. Phylogenetic Analysis, Paralogon Groups, and Fingerprints

Robert Fredriksson, Malin C. Lagerström, Lars‐Gustav Lundin et al. · Molecular Pharmacology · 2003 · 2.9K citations

A ternary complex model explains the agonist-specific binding properties of the adenylate cyclase-coupled beta-adrenergic receptor.

A. De Léan, Jeffrey M. Stadel, Robert J. Lefkowitz · Journal of Biological Chemistry · 1980 · 1.6K citations · Full text

Agonist-specific Binding Properties, Experimental Pharmacology, Ternary Complex Hrx +17

Crystal structure of opsin in its G-protein-interacting conformation

Patrick Scheerer, Jung Hee Park, Peter W. Hildebrand et al. · Nature · 2008 · 1K citations

Crystal Structure, Protein X-ray Crystallography, Structural Biology +1