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Pre-clinical characterization of aryloxypyridine amides as histamine H3 receptor antagonists: Identification of candidates for clinical development

Michael A. Letavic, Leah Aluisio, John Atack, Pascal Bonaventure, Nicholas I. Carruthers, Christine Dugovic, Anita Everson, Mark A. Feinstein, Ian Fraser, Kenway Hoey,

Bioorganic & Medicinal Chemistry Letters · 2010 · 27 citations · 5 references

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5

Acute wake‐promoting actions of JNJ‐5207852, a novel, diamine‐based H<sub>3</sub> antagonist

Ann Barbier, Craig W. Berridge, Christine Dugovic et al. · British Journal of Pharmacology · 2004 · 143 citations · Full text

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A New Class of Diamine-Based Human Histamine H<sub>3</sub> Receptor Antagonists:  4-(Aminoalkoxy)benzylamines

Richard L. Apodaca, Curt A. Dvorak, Wei Xiao et al. · Journal of Medicinal Chemistry · 2003 · 119 citations · Full text

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Microwave assisted, palladium catalyzed aminocarbonylations of heteroaromatic bromides using solid Mo(CO)6 as the carbon monoxide source

Michael A. Letavic, Kiev S. Ly · Tetrahedron Letters · 2007 · 48 citations

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Synthesis and biological activity of piperazine and diazepane amides that are histamine H3 antagonists and serotonin reuptake inhibitors

Kiev S. Ly, Michael A. Letavic, John M. Keith et al. · Bioorganic & Medicinal Chemistry Letters · 2007 · 26 citations · Full text

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Diamine-based human histamine H3 receptor antagonists: (4-Aminobutyn-1-yl)benzylamines

Curt A. Dvorak, Richard L. Apodaca, Wei Xiao et al. · European Journal of Medicinal Chemistry · 2009 · 12 citations · Full text

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