Concepedia

Initial structure–activity relationships of lysophosphatidic acid receptor antagonists: discovery of a high-affinity LPA1/LPA3 receptor antagonist

Brian Heasley, Renata Jarosz, Kevin R. Lynch, Timothy L. Macdonald

Bioorganic & Medicinal Chemistry Letters · 2004 · 61 citations · 9 references

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References

9

Identification of p2y9/GPR23 as a Novel G Protein-coupled Receptor for Lysophosphatidic Acid, Structurally Distant from the Edg Family

Kyoko Noguchi, Satoshi Ishii, Takao Shimizu · Journal of Biological Chemistry · 2003 · 557 citations · Full text

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Identification of an intracellular receptor for lysophosphatidic acid (LPA): LPA is a transcellular PPARγ agonist

Thomas M. McIntyre, Aaron V. Pontsler, Adriana Ribeiro Silva et al. · Proceedings of the National Academy of Sciences · 2002 · 545 citations · Full text

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Characterization of an ovarian cancer activating factor in ascites from ovarian cancer patients.

Yan Xu, Douglas C. Gaudette, Jessica Boynton et al. · PubMed · 1995 · 324 citations

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Molecular Cloning and Characterization of a Lysophosphatidic Acid Receptor, Edg-7, Expressed in Prostate

Dong‐Soon Im, Christopher E. Heise, Michael A. Harding et al. · Molecular Pharmacology · 2000 · 199 citations

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Phenotypic Modulation of Vascular Smooth Muscle Cells Induced by Unsaturated Lysophosphatidic Acids

Ken’ichiro Hayashi, Masanori Takahashi, Wataru Nishida et al. · Circulation Research · 2001 · 192 citations · Full text

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