Concepedia

Structure–activity relationships of 3,5-disubstituted benzamides as glucokinase activators with potent in vivo efficacy

Tomoharu Iino, Noriaki Hashimoto, Kaori Sasaki, Sumika Ohyama, Riki Yoshimoto, Hideka Hosaka, Takuro Hasegawa, Masato Chiba, Yasufumi Nagata, Jun‐ichi Eiki,

Bioorganic & Medicinal Chemistry · 2009 · 50 citations · 16 references

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16

New N- and O-arylations with phenylboronic acids and cupric acetate

Dominic M. T. Chan, Kevin L. Monaco, Ru-Ping Wang et al. · Tetrahedron Letters · 1998 · 1.1K citations

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When poor solubility becomes an issue: From early stage to proof of concept

Sven Stegemann, F. Leveiller, D. Franchi et al. · European Journal of Pharmaceutical Sciences · 2007 · 504 citations

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Structural Basis for Allosteric Regulation of the Monomeric Allosteric Enzyme Human Glucokinase

Kenji Kamata, Morihiro Mitsuya, T. Nishimura et al. · Structure · 2004 · 503 citations · Full text

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When poor solubility becomes an issue: from early stage to proof of concept

Sven Stegemann · 2007 · 390 citations

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Banting Lecture 1995. A lesson in metabolic regulation inspired by the glucokinase glucose sensor paradigm

Franz M. Matschinsky · Diabetes · 1996 · 154 citations

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