Agonist and Inverse Agonist Efficacy at Human Recombinant Serotonin 5-HT 1A Receptors as a Function of Receptor:G-protein Stoichiometry

A JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS

Journal of the American Medical Association · 1909 · 7.9K citations · Full text

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The genomic clone G-21 which resembles a β-adrenergic receptor sequence encodes the 5-HT1A receptor

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Antagonists with negative intrinsic activity at delta opioid receptors coupled to GTP-binding proteins.

Tommaso Costa, A. Herz · Proceedings of the National Academy of Sciences · 1989 · 530 citations · Full text

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Electrophysiological, biochemical, neurohormonal and behavioural studies with WAY-100635, a potent, selective and silent 5-HT1A receptor antagonist

Allan Fletcher, Elaine A. Forster, David J. Bill et al. · Behavioural Brain Research · 1995 · 521 citations

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Modulation by mu-opioid agonists of guanosine-5'-O-(3-[35S]thio)triphosphate binding to membranes from human neuroblastoma SH-SY5Y cells.

John R. Traynor, Stefan R. Nahorski · Molecular Pharmacology · 1995 · 462 citations

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