Concepedia

Synthesis, biological evaluation, and molecular modeling studies of new 1,3,4-oxadiazole- and 1,3,4-thiadiazole-substituted 4-oxo-4H-pyrido[1,2-a]pyrimidines as anti-HIV-1 agents

Zahra Hajimahdi, Afshin Zarghi, Rezvan Zabihollahi, Mohammad Reza Aghasadeghi

Medicinal Chemistry Research · 2012 · 64 citations · 15 references

DOI

Concepts

References

15

Automated docking using a Lamarckian genetic algorithm and an empirical binding free energy function

Garrett M. Morris, David S. Goodsell, Robert S. Halliday et al. · Journal of Computational Chemistry · 1998 · 10.8K citations

, , +17

Evaluation of a soluble tetrazolium/formazan assay for cell growth and drug sensitivity in culture using human and other tumor cell lines.

Dominic A. Scudiero, Robert H. Shoemaker, Kenneth D. Paull et al. · PubMed · 1988 · 2.4K citations

, , +9

5-Substituted-1H-tetrazoles as carboxylic acid isosteres: medicinal chemistry and synthetic methods

R. Jason Herr · Bioorganic & Medicinal Chemistry · 2002 · 844 citations

, , +13

5‐Substituted 1H‐Tetrazoles as Carboxylic Acid Isosteres: Medicinal Chemistry and Synthetic Methods

R. Jason Herr · ChemInform · 2003 · 681 citations

, , +15

Retroviral intasome assembly and inhibition of DNA strand transfer

S. Hare, Saumya Gupta, Eugene Valkov et al. · Nature · 2010 · 666 citations · Full text

, , +13