The synthesis of amino-acid functionalized β-Carbolines as topoisomerase II inhibitors

Total Synthesis of Baccatin III and Taxol

Samuel J. Danishefsky, John J. Masters, Wendy B. Young et al. · Journal of the American Chemical Society · 1996 · 429 citations

Diversity Oriented Synthesis, Bioorganic Chemistry, Engineering +14

Novel Mammalian Cell Cycle Inhibitors, Tryprostatins A, B and Other Diketopiperazines Produced by Aspergillus fumigatus. I. Taxonomy, Fermentation, Isolation and Biological Properties.

Cheng‐Bin Cui, Hideaki Kakeya, Gen Okada et al. · The Journal of Antibiotics · 1996 · 208 citations · Full text

Enantiospecific Formation of <i>Trans</i> 1,3-Disubstituted Tetrahydro-β-carbolines by the Pictet−Spengler Reaction and Conversion of <i>Cis</i> Diastereomers into Their <i>Trans</i> Counterparts by Scission of the C-1/N-2 Bond

Eric Cox, Linda K. Hamaker, Jin Li et al. · The Journal of Organic Chemistry · 1997 · 103 citations

Trans Diastereomers, Enantioselective Synthesis, Engineering +15

Total Synthesis of Tryprostatin B:  Generation of a Nucleophilic Prenylating Species from a Prenylstannane

Kristopher M. Depew, Samuel J. Danishefsky, Neal Rosen et al. · Journal of the American Chemical Society · 1996 · 84 citations

Bioorganic Chemistry, Engineering, Altmetric Attention Score +16

Antitumor Agents. 163. Three-Dimensional Quantitative Structure−Activity Relationship Study of 4‘-<i>O</i>-Demethylepipodophyllotoxin Analogs Using the Modified CoMFA/q²-GRS Approach

Sung Jin Cho, Alexander Tropsha, Matthew Suffness et al. · Journal of Medicinal Chemistry · 1996 · 81 citations