Synthetic Communications · 1975 · 49 citations · 6 references
Natural SciencesChemistryMedicinal ChemistryOrganic ChemistrySynthetic Medicinal ChemistryHeterocycle SynthesisHeterocyclic ChemistryHeterocyclic CompoundsOrganic SynthesisAzetidine ChemistryHeterocyclic Medicinal ChemistryMedicinal Heterocycles
Abstract In spite of the fact that a number of methods are available for the preparation of aziridines, general synthetic routes leading to 1,2-disubstituted aziridines remained laborious in most cases(2-6). A convenient and versatile synthesis is desirable in order to permit studies of this important biologically active heterocyclic system.
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