Publication | Open Access

Thieno[2,3-b]pyridines as negative allosteric modulators of metabotropic GluR5 receptors: Hit-to-lead optimization

Negative Allosteric ModulatorsBiochemistryFunctional SelectivityMetabotropic Glur5 ReceptorsMedicineG Protein-coupled ReceptorReceptor (Biochemistry)Mechanism Of ActionPharmacological AgentHit-to-lead OptimizationPharmacotherapyPharmacologyDrug Discovery