Concepedia

One-Pot Synthesis of Azaindoles via Palladium-Catalyzed α-Heteroarylation of Ketone Enolates

Steven H. Spergel, Danielle R. Okoro, William J. Pitts

The Journal of Organic Chemistry · 2010 · 36 citations · 24 references

DOI

Concepts

Abstract

A convenient, one-pot method for the construction of a variety of azaindoles using simple ketones and haloaminopyridines is described.

References

24

Well-Defined N-Heterocyclic Carbenes−Palladium(II) Precatalysts for Cross-Coupling Reactions

Nicolas Marion, Steven P. Nolan · Accounts of Chemical Research · 2008 · 1K citations

, , +15

Palladium-Catalyzed α-Arylation of Carbonyl Compounds and Nitriles

Darcy A. Culkin, John F. Hartwig · Accounts of Chemical Research · 2003 · 934 citations

, , +12

Synthesis of indoles via palladium-catalyzed heteroannulation of internal alkynes

Richard C. Larock · Journal of the American Chemical Society · 1991 · 824 citations

, , +11

Highly Active and Selective Catalysts for the Formation of α-Aryl Ketones

Joseph M. Fox, Xiaohua Huang, A. Chieffi et al. · Journal of the American Chemical Society · 2000 · 517 citations

, , +16

Direct C−H Bond Arylation:  Selective Palladium-Catalyzed C2-Arylation of <i>N</i>-Substituted Indoles

Benjamin S. Lane, Dalibor Sameš · Organic Letters · 2004 · 261 citations

, , +17