An efficient synthesis of 2,3-diaryl (3H)-quinazolin-4-ones via imidoyl chlorides

Synthesis and biological evaluation of 2-styrylquinazolin-4(3H)-ones, a new class of antimitotic anticancer agents which inhibit tubulin polymerization

Jack B. Jiang, David P. Hesson, Betsy A. Dusak et al. · Journal of Medicinal Chemistry · 1990 · 261 citations

Medicine, Medicinal Chemistry, Pharmacology +14

Quinazolinone Derivatives as Orally Available Ghrelin Receptor Antagonists for the Treatment of Diabetes and Obesity

Joachim Rudolph, William P. Esler, Stephen O’Connor et al. · Journal of Medicinal Chemistry · 2007 · 157 citations · Full text

Medicine, Endocrinology, Pharmacology +17

Palladium-Catalyzed Cyclocarbonylation of <i>o</i>-Iodoanilines with Heterocumulenes:  Regioselective Preparation of 4(3<i>H</i>)-Quinazolinone Derivatives

Chitchamai Larksarp, Howard Alper · The Journal of Organic Chemistry · 2000 · 153 citations

Natural Sciences, Chemistry, Medicinal Chemistry +16

New Type of Febrifugine Analogues, Bearing a Quinolizidine Moiety, Show Potent Antimalarial Activity against <i>Plasmodium</i> Malaria Parasite

Yoshiaki Takaya, Hidehisa Tasaka, Tomoyuki Chiba et al. · Journal of Medicinal Chemistry · 1999 · 139 citations

Medicine, Medicinal Chemistry, Pharmacology +15

Microwave-assisted one-pot synthesis of 2,3-disubstituted 3H-quinazolin-4-ones

Jifeng Liu, Jaekyoo Lee, Audra M. Dalton et al. · Tetrahedron Letters · 2005 · 137 citations

Natural Sciences, Chemistry, Medicinal Chemistry +11