Concepedia

Discovery of novel A3 adenosine receptor ligands based on chromone scaffold

Alexandra Gaspar, Joana Reis, Sonja Kachler, Silvia Paoletta, Eugenio Uriarte, Karl‐Norbert Klotz, Stefano Moro, Fernanda Borges

Biochemical Pharmacology · 2012 · 47 citations · 16 references

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16

Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

Yung-Chi Cheng, William H. Prusoff · Biochemical Pharmacology · 1973 · 12.9K citations

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Glide:  A New Approach for Rapid, Accurate Docking and Scoring. 1. Method and Assessment of Docking Accuracy

Richard A. Friesner, Jay L. Banks, Robert B. Murphy et al. · Journal of Medicinal Chemistry · 2004 · 9.9K citations

, , +17

The 2.6 Angstrom Crystal Structure of a Human A <sub>2A</sub> Adenosine Receptor Bound to an Antagonist

Veli‐Pekka Jaakola, Mark T. Griffith, Michael A. Hanson et al. · Science · 2008 · 1.8K citations · Full text

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Empirical Scoring Functions for Advanced Protein−Ligand Docking with PLANTS

Oliver Korb, Thomas Stützle, Thomas E. Exner · Journal of Chemical Information and Modeling · 2009 · 1.3K citations

, , +14

Recent development of peptide coupling reagents in organic synthesis

So‐Yeop Han, Young‐Ah Kim · Tetrahedron · 2004 · 756 citations

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