Journal of Pharmacology and Experimental Therapeutics · 1991 · 112 citations · 0 references
PharmacyChemistryPharmacologyDrug DiscoveryOrganic ChemistryStructure-activity RelationshipsDrug-receptor InteractionsLigand BindingPotency OptimizationReceptor PharmacologyReceptor-ligand InteractionsStructure-activity Relationship AnalysisCompound Potency OptimizationLigand ChemistryMedicinal Chemistry ApplicationsReceptor Binding AssaysReceptor Selectivity ProfilingReceptorsRing Size Effects