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Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

Yung-Chi Cheng, William H. Prusoff · Biochemical Pharmacology · 1973 · 12.9K citations

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J.M. Baldwin · The EMBO Journal · 1993 · 979 citations · Full text

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Gebhard F. X. Schertler, Claudio Villa, Richard A. Henderson · Nature · 1993 · 760 citations

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An alpha-carbon template for the transmembrane helices in the rhodopsin family of G-protein-coupled receptors 1 1Edited by R. Huber

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