Concepedia

Synthesis of new fluorinated analogs of GABA, Pregabalin bioisosteres, and their effects on [3H]GABA uptake by rat brain nerve terminals

Natalia Pozdnyakova, Elena N. Shaitanova, Igor I. Gerus, Marina Dudarenko, Roman V. Mironets, Günter Haufe, Valery P. Kukhar

Bioorganic & Medicinal Chemistry · 2015 · 17 citations · 28 references

DOI

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References

28

Fluorine in medicinal chemistry: Recent therapeutic applications of fluorinated small molecules

Kenneth L. Kirk · Journal of Fluorine Chemistry · 2006 · 892 citations

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Organofluorine compounds in medicinal chemistry and biomedical applications

International Journal of Biochemistry · 1994 · 489 citations

, , +7

Artificial reductant enhancement of the Lowry method for protein determination

Eric M. Larson, Bruce Howlett, André T. Jagendorf · Analytical Biochemistry · 1986 · 326 citations

, , +5

Structure−Activity Relationships of Pregabalin and Analogues That Target the α<sub>2</sub>-δ Protein

Thomas R. Belliotti, Thomas Capiris, I. Victor Ekhato et al. · Journal of Medicinal Chemistry · 2005 · 210 citations

, , +17

From Basic Science to Blockbuster Drug: The Discovery of Lyrica

Richard B. Silverman · Angewandte Chemie International Edition · 2008 · 167 citations

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