Concepedia
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Publications
4
Citations
140
Authors
3
Location
Cambridge, United Kingdom
Cypralis (United Kingdom) is a company institution in Cambridge, United Kingdom known for pharmacology, medicinal chemistry, and drug discovery.
Top concepts
PharmacyDrug DesignPharmacologyDrug DiscoveryLead OptimizationMedicinal ChemistryMacrocyclic InhibitorsMacrocyclic Drug Designπ StackingLigand Binding
Cypralis (United Kingdom), United Kingdom
12 publications · 2.7K citations
6
h-index
3 publications · 180 citations
2 publications · 87 citations
2
1–3 of 3
Discovery of a Potent and Orally Bioavailable Cyclophilin Inhibitor Derived from the Sanglifehrin Macrocycle
Richard L. Mackman, Victoria A. Steadman, David K. Dean et al. · Journal of Medicinal Chemistry · 2018 · 78 citations · Full text
Pharmacy, Medicinal Chemistry, Pharmacology +17
Discovery of Potent Cyclophilin Inhibitors Based on the Structural Simplification of Sanglifehrin A
Victoria A. Steadman, S. Pettit, Karine G. Poullennec et al. · Journal of Medicinal Chemistry · 2017 · 58 citations · Full text
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