Selective Receptor Modulation
Selective Receptor Modulation is a pharmacological mechanism in which a ligand differentially activates or inhibits a steroid hormone receptor in a tissue-specific or context-dependent manner, thereby producing selective agonistic or antagonistic effects distinct from full agonists or antagonists.
108
Publications
5.6K
Citations
605
Authors
232
Institutions
Publications per year
2017–2026
13
Parents
108
Derivatives of Erythropoietin That Are Tissue Protective But Not Erythropoietic
Marcel Leist, Pietro Ghezzi, Giovanni Grasso et al. · Science · 2004 · 798 citations · Full text
Medicine, Neuroscience, Pharmacology +14
Differential Targeting of Gßγ-Subunit Signaling with Small Molecules
Tabetha M. Bonacci, Jennifer Mathews, Chujun Yuan et al. · Science · 2006 · 231 citations
1–5 of 108
605
Centre National de la Recherche Scientifique, France
2 publications · 58 citations
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2
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1–5 of 605
232
Eli Lilly (United States)
Indianapolis, United States
3 h-index
9 publications
277 citations
Université de Strasbourg
Strasbourg, France
2 h-index
12 publications
348 citations
Duke University
Durham, United States
2 h-index
7 publications
183 citations
GlaxoSmithKline (United States)
Philadelphia, United States
2 h-index
6 publications
162 citations

GlaxoSmithKline (United Kingdom)
London, United Kingdom
2 h-index
6 publications
162 citations
Inserm
Paris, France
2 h-index
17 publications
607 citations

University of Leicester
Leicester, United Kingdom
2 h-index
5 publications
112 citations

Howard Hughes Medical Institute
Chevy Chase, United States
2 h-index
6 publications
213 citations
1–8 of 232
Repository · 5 publications · 250 citations
5
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EJP · 5 publications · 142 citations
5
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4 publications · 1.7K citations
4
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3 publications · 104 citations
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JI · 3 publications · 68 citations
3
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1–5