Metal-free hydroacyloxylation and hydration reactions of ynamides: synthesis of α-acyloxyenamides and N-acylsulfonamides

Shijie Xu, Jian‐Quan Liu, Donghua Hu, +1

Green Chemistry

Chemical EngineeringMetal-free ConditionsDerivativesEngineeringDerivative (Chemistry) +11

Identification of benzothiazinones containing an oxime functional moiety as new anti-tuberculosis agents

Apeng Wang, Kai Lv, Zeyu Tao, +11

European Journal of Medicinal Chemistry

New Anti-tuberculosis AgentsOxime Functional MoietyBioorganic ChemistryHeterocyclicBiochemistry +7

Design, synthesis and biological activity of N-(amino)piperazine-containing benzothiazinones against Mycobacterium tuberculosis

Apeng Wang, Shijie Xu, Yun Chai, +9

European Journal of Medicinal Chemistry

Biological ActivityPiperazine-containing BenzothiazinonesMedicineDrug DiscoveryMycobacterium Tuberculosis +5

Palladium-catalyzed one-pot cycloaddition reactions of thioureas with 3<i>H</i>-indol-3-ones generated<i>in situ</i>from 2-alkynyl arylazides: rapid and efficient access to imidazoloindolines

Ping Li, Boyu Zhu, Yao Xu, +5

Organic Chemistry Frontiers

Cross-coupling ReactionEngineeringOrganic Chemistry2-Alkynyl ArylazidesCatalysis +8

PPh₃-Mediated Cascade Reaction of 2-Alkynylnitrobenzenes and Thioureas for the Construction of Imidazo[4,5-<i>b</i>]indole-2-thiones

Yao Xu, Hui Fan, Fan Yang, +4

The Journal of Organic Chemistry

DBN‐Catalyzed Regioselective Acylation of Carbohydrates and Diols in Ethyl Acetate

Bo Ren, Mengyao Zhang, Shijie Xu, +3

European Journal of Organic Chemistry

Selective AcylationEngineeringNatural SciencesBiocatalysisOrganic Chemistry +9

Optimization and SAR research at the piperazine and phenyl rings of JNJ4796 as new anti-influenza A virus agents, part 1

Aoyu Wang, Yuhuan Li, Kai Lv, +10

European Journal of Medicinal Chemistry

Part 1Phenyl RingsAntiviral Drug DevelopmentSar ResearchInfluenza Vaccine +3

Design, synthesis and biological evaluation of nitrofuran-1,3,4-oxadiazole hybrids as new antitubercular agents

Apeng Wang, Shijie Xu, Yun Chai, +9

Bioorganic & Medicinal Chemistry

Combinatorial ChemistryBioorganic ChemistryMedicineNew Antitubercular AgentsBiological Evaluation +6

PPh₃‐Mediated Wittig‐Like/Mannich Tandem Reactions of 2‐Alkynylnitrobenzenes with Ketones for the Synthesis of 2,2‐Disubstituted Indolin‐3‐Ones

Hui Fan, Yao Xu, Fan Yang, +3

Advanced Synthesis & Catalysis

Mannich AdditionDiversity Oriented SynthesisDerivativesWittig‐like/mannich Tandem ReactionsEngineering +11

Design, synthesis and antimycobacterial activity of new benzothiazinones inspired by rifampicin/rifapentine

Apeng Wang, Yu Lu, Kai Lv, +6

Bioorganic Chemistry

Medicinal ChemistryNatural Product SynthesisPharmaceutical ChemistryMedicineAntibacterial Agent +8