Concepedia

Palladium-catalyzed one-pot cycloaddition reactions of thioureas with 3<i>H</i>-indol-3-ones generated<i>in situ</i>from 2-alkynyl arylazides: rapid and efficient access to imidazoloindolines

Ping Li, Boyu Zhu, Yao Xu, Zhiqiang Zhou, Guiwen Hu, Fan Yang, Shijie Xu, Xiaoxiang Zhang

Organic Chemistry Frontiers · 2020 · 21 citations · 59 references

DOI

Concepts

Abstract

An efficient palladium-catalyzed one-pot synthesis of imidazoloindolines from 2-alkynyl arylazides under mild reaction conditions has been described.

References

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