Amitgiri Goswami

Diaryl Dihydropyrazole-3-carboxamides with Significant In Vivo Antiobesity Activity Related to CB1 Receptor Antagonism:  Synthesis, Biological Evaluation, and Molecular Modeling in the Homology Model

Brijesh Kumar Srivastava, Amit Joharapurkar, Saurin Raval et al. · Journal of Medicinal Chemistry · 2007 · 64 citations · Full text

Lead Compounds, Pharmaceutical Science, Drug Target +19

Revisiting glitazars: Thiophene substituted oxazole containing α-ethoxy phenylpropanoic acid derivatives as highly potent PPARα/γ dual agonists devoid of adverse effects in rodents

Preeti Raval, Mukul Jain, Amitgiri Goswami et al. · Bioorganic & Medicinal Chemistry Letters · 2011 · 22 citations · Full text

Molecular Pharmacology, Pharmacological Study, Physiology +7

Discovery of a highly orally bioavailable c-5-[6-(4-Methanesulfonyloxyphenyl)hexyl]-2-methyl-1,3-dioxane-r-2-carboxylic acid as a potent hypoglycemic and hypolipidemic agent

Harikishore Pingali, Mukul R. Jain, Shailesh R. Shah et al. · Bioorganic & Medicinal Chemistry Letters · 2008 · 14 citations · Full text

Medicinal Chemistry, Pharmaceutical Science, Biochemistry +9

Bioisosteric replacement of dihydropyrazole of 4S-(−)-3-(4-chlorophenyl)-N-methyl-N′-[(4-chlorophenyl)-sulfonyl]-4-phenyl-4,5-dihydro-1H-pyrazole-1-caboxamidine (SLV-319) a potent CB1 receptor antagonist by imidazole and oxazole

Brijesh Kumar Srivastava, Rina Soni, Amit Joharapurkar et al. · Bioorganic & Medicinal Chemistry Letters · 2007 · 13 citations

Bioisosteric Replacement, Molecular Pharmacology, Bioorganic Chemistry +10

Convenient Synthesis of Structurally Novel 1,3‐Disubstituted Azetidine Derivatives

Rajendra K. Kharul, Amitgiri Goswami, Archana Gite et al. · Synthetic Communications · 2008 · 10 citations

Derivatives, Core Structure, Azetidine Building Block +5