Kousei Yoshihara

Synthetic studies on polypropionate antibiotics based on the stereospecific methylation of γ δ-epoxy acrylates by trimethylaluminum. A highly stereoselective construction of the eight contiguous chiral centers of ansa-chains of rifamycins

Masaaki Miyashita, Kousei Yoshihara, Katsumi Kawamine et al. · Tetrahedron Letters · 1993 · 29 citations

Medicinal Chemistry, Engineering, Organic Chemistry +10

Synthesis and SAR study of new thiazole derivatives as vascular adhesion protein-1 (VAP-1) inhibitors for the treatment of diabetic macular edema

Takayuki Inoue, Masataka Morita, Takashi Tojo et al. · Bioorganic & Medicinal Chemistry · 2012 · 25 citations · Full text

Ophthalmology, Medicine, Vascular Pharmacology +8

Gas-sensing properties of semiconductor heterolayers fabricated by a slide-off transfer printing method

Akihiko KAWAHARA, Kousei Yoshihara, Hiroaki Katsuki et al. · Sensors and Actuators B Chemical · 2000 · 24 citations

Materials Science, Engineering, Gas Sensor +8

A stereocontrolled enantiospecific route to tirandamycin B

Tomonori Shiratani, Kiyoshi Kimura, Kousei Yoshihara et al. · Chemical Communications · 1996 · 17 citations

δ-Epoxy Acrylate 5, Medicinal Chemistry, Bioorganic Chemistry +15

Discovery and biological evaluation of novel pyrazolopyridine derivatives as potent and orally available PI3Kδ inhibitors

Toshihiro Hamajima, Fumie Takahashi, Koji Kato et al. · Bioorganic & Medicinal Chemistry · 2018 · 15 citations · Full text

Medicinal Chemistry, Biochemistry, Novel Pyrazolopyridine Derivatives +11