New α-(N)-heterocyclichydrazones: evaluation of anticancer, anti-HIV and antimicrobial activity

Luisa Savini, Luisa Chiasserini, Valter Travagli, +4

European Journal of Medicinal Chemistry

Medicinal ChemistryBiochemistryMedicineNew α-Natural Sciences +5

Synthesis of N1-arylidene-N2-quinolyl- and N2-acrydinylhydrazones as potent antimalarial agents active against CQ-resistant P. falciparum strains

Sandra Gemma, Gagan Kukreja, Caterina Fattorusso, +10

Bioorganic & Medicinal Chemistry Letters

Antiparasitic AgentMedicineMalariaAntimicrobial ChemotherapyPotent Antimalarial Agents +3

Specific Targeting of Acetylcholinesterase and Butyrylcholinesterase Recognition Sites. Rational Design of Novel, Selective, and Highly Potent Cholinesterase Inhibitors

Luisa Savini, Alessandra Gaeta, Caterina Fattorusso, +7

Journal of Medicinal Chemistry

Butyrylcholinesterase Recognition SitesDrug TargetBioorganic ChemistryChemical BiologyPharmaceutical Chemistry +15

Synthesis and anti-tubercular evaluation of 4-quinolylhydrazones

Luisa Savini, Luisa Chiasserini, Alessandra Gaeta, +1

Bioorganic & Medicinal Chemistry

PharmacologyAnti-tubercular EvaluationStereoselective SynthesisNatural Product Synthesis

Design, Synthesis, and Structure–Activity Relationship Studies of 4-Quinolinyl- and 9-Acrydinylhydrazones as Potent Antimalarial Agents

Caterina Fattorusso, Giuseppe Campiani, Gagan Kukreja, +17

Journal of Medicinal Chemistry

Specific Targeting of Hepatitis C Virus NS3 RNA Helicase. Discovery of the Potent and Selective Competitive Nucleotide-Mimicking Inhibitor QU663

Giovanni Maga, Sandra Gemma, Caterina Fattorusso, +11

Biochemistry

Structural study of ribonucleotide reductase inhibitor hydrazones. Synthesis and X-ray diffraction analysis of a copper(II)-benzoylpyridine-2-quinolinyl hydrazone complex

Gabriella Tamasi, Luisa Chiasserini, Luisa Savini, +2

Journal of Inorganic Biochemistry

Inorganic CompoundBiochemistryStructure ElucidationStructural StudyX-ray Diffraction Analysis +2

Mimicking the Intramolecular Hydrogen Bond: Synthesis, Biological Evaluation, and Molecular Modeling of Benzoxazines and Quinazolines as Potential Antimalarial Agents

Sandra Gemma, Caterina Camodeca, Margherita Brindisi, +21

Journal of Medicinal Chemistry

Combinatorial ChemistryBioorganic ChemistryAntiparasitic AgentMalariaOrganic Chemistry +15

Pyrroloquinoxaline hydrazones as fluorescent probes for amyloid fibrils

Sandra Gemma, Laura Colombo, Gianluigi Forloni, +13

Organic & Biomolecular Chemistry

Development of Molecular Probes for the Identification of Extra Interaction Sites in the Mid-Gorge and Peripheral Sites of Butyrylcholinesterase (BuChE). Rational Design of Novel, Selective, and Highly Potent BuChE Inhibitors

Giuseppe Campiani, Caterina Fattorusso, Stefania Butini, +13

Journal of Medicinal Chemistry

Drug TargetBioorganic ChemistryOrganic ChemistryChemical BiologyPharmaceutical Chemistry +19