Ya-Qiu Long

Rational Design and Synthesis of Novel Dimeric Diketoacid-Containing Inhibitors of HIV-1 Integrase:  Implication for Binding to Two Metal Ions on the Active Site of Integrase

Ya-Qiu Long, Xiao-Hua Jiang, Raveendra Dayam et al. · Journal of Medicinal Chemistry · 2004 · 179 citations · Full text

Targeting Inactive Enzyme Conformation: Aryl Diketoacid Derivatives as a New Class of PTP1B Inhibitors

Sijiu Liu, Li‐Fan Zeng, Wu Li et al. · Journal of the American Chemical Society · 2008 · 83 citations · Full text

Drug Target, Molecular Biology, Chemical Biology +16

Design and discovery of flavonoid-based HIV-1 integrase inhibitors targeting both the active site and the interaction with LEDGF/p75

Bo-Wen Li, Feng-Hua Zhang, Erik Serrao et al. · Bioorganic & Medicinal Chemistry · 2014 · 58 citations · Full text

Medicinal Chemistry, Biochemistry, Medicine +10

Repositioning HIV-1 Integrase Inhibitors for Cancer Therapeutics: 1,6-Naphthyridine-7-carboxamide as a Promising Scaffold with Drug-like Properties

Li‐Fan Zeng, Yong Wang, Roza Kazemi et al. · Journal of Medicinal Chemistry · 2012 · 55 citations · Full text

Combinatorial Chemistry, Hiv-1 Integrase, Bioorganic Chemistry +18

Discovery of a Novel Nonphosphorylated Pentapeptide Motif Displaying High Affinity for Grb2-SH2 Domain by the Utilization of 3‘-Substituted Tyrosine Derivatives

Yan-Li Song, Megan L. Peach, Peter P. Roller et al. · Journal of Medicinal Chemistry · 2006 · 48 citations · Full text