Gregory Ciszewski

Discovery of Pyrano[3,4-<i>b</i>]indoles as Potent and Selective HCV NS5B Polymerase Inhibitors

Ariamala Gopalsamy, Kitae Lim, Gregory Ciszewski et al. · Journal of Medicinal Chemistry · 2004 · 96 citations · Full text

Replicon System, Novel Series, Biochemistry +12

Discovery of Proline Sulfonamides as Potent and Selective Hepatitis C Virus NS5b Polymerase Inhibitors. Evidence for a New NS5b Polymerase Binding Site

Ariamala Gopalsamy, Rajiv Chopra, Kitae Lim et al. · Journal of Medicinal Chemistry · 2006 · 52 citations · Full text

Crystal Structure, Bioorganic Chemistry, Molecular Biology +19

Synthesis of Pyrazolo[1,5-α]pyrimidinone Regioisomers

Lori K. Gavrin, Arthur Lee, Brian A. Provencher et al. · The Journal of Organic Chemistry · 2006 · 49 citations

Design and synthesis of 3,4-dihydro-1H-[1]-benzothieno[2,3-c]pyran and 3,4-dihydro-1H-pyrano[3,4-b]benzofuran derivatives as non-nucleoside inhibitors of HCV NS5B RNA dependent RNA polymerase

Ariamala Gopalsamy, Alexis Aplasca, Gregory Ciszewski et al. · Bioorganic & Medicinal Chemistry Letters · 2005 · 39 citations · Full text

Medicine, Drug Discovery, Non-nucleoside Inhibitors +4

Late-Stage Lead Diversification Coupled with Quantitative Nuclear Magnetic Resonance Spectroscopy to Identify New Structure–Activity Relationship Vectors at Nanomole-Scale Synthesis: Application to Loratadine, a Human Histamine H ₁ Receptor Inverse Agonist

Manjinder S. Lall, Asser Bassyouni, James Bradow et al. · Journal of Medicinal Chemistry · 2020 · 30 citations · Full text