Concepedia
7
Publications
1.8K
Citations
H-Index
2008
Active since
Affiliations
Portland VA Medical Center(Current)
Oregon Health & Science University
Brigham and Women's Hospital
Dana-Farber Cancer Institute
Harvard University
Arin McKinley is an author at Portland VA Medical Center specializing in drug discovery, systems biology, and tumor biology.
Top concepts
MedicinePharmacologyTumor BiologyDrug DiscoverySystems Biology
Publications per year
2008–2019
Primary and Secondary Kinase Genotypes Correlate With the Biological and Clinical Activity of Sunitinib in Imatinib-Resistant Gastrointestinal Stromal Tumor
Michael C. Heinrich, Robert G. Maki, Christopher L. Corless et al. · Journal of Clinical Oncology · 2008 · 799 citations · Full text
Ripretinib (DCC-2618) Is a Switch Control Kinase Inhibitor of a Broad Spectrum of Oncogenic and Drug-Resistant KIT and PDGFRA Variants
Bryan D. Smith, Michael D. Kaufman, Wei-Ping Lu et al. · Cancer Cell · 2019 · 270 citations
Pdgfra Variants, Oncogenic Agent, Medicine +9
Crenolanib Inhibits the Drug-Resistant PDGFRA D842V Mutation Associated with Imatinib-Resistant Gastrointestinal Stromal Tumors
Michael C. Heinrich, Diana Griffith, Arin McKinley et al. · Clinical Cancer Research · 2012 · 218 citations
Phase II, Open-Label Study Evaluating the Activity of Imatinib in Treating Life-Threatening Malignancies Known to Be Associated with Imatinib-Sensitive Tyrosine Kinases
Michael C. Heinrich, Heikki Joensuu, George D. Demetri et al. · Clinical Cancer Research · 2008 · 212 citations
Complementary activity of tyrosine kinase inhibitors against secondary kit mutations in imatinib-resistant gastrointestinal stromal tumours
César Serrano, Adrián Mariño‐Enríquez, Derrick L. Tao et al. · British Journal of Cancer · 2019 · 159 citations · Full text
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