Time-resolved FRET between GPCR ligands reveals oligomers in native tissues

Laura Albizu, Martin Cottet, Michaela Králíková, +16

Nature Chemical Biology

Signal TransductionMolecular PhysiologyG Protein-coupled ReceptorNatural SciencesReceptor (Biochemistry) +9

Molecular pharmacology of AVP and OT receptors and therapeutic potential

Claude Barberis, Didier Morin, Thierry Durroux, +6

Drug News & Perspectives

Molecular PharmacologyAllergyMedicineReceptor (Biochemistry)Neuropeptide Receptor +3

IMMUNOLOGIC IDENTIFICATION OF BOTH PLASMA AND HUMAN RENAL INACTIVE RENIN AS PRORENIN

J Bouhnik, Jean‐Alain Fehrentz, F. X. Galen, +5

The Journal of Clinical Endocrinology & Metabolism

Peptide Coupling Reagents; VIII. A High Yield Preparation of Phenyl Esters of Amino Acids using Benzotriazolyloxytris[dimethylamino]phosphonium Hexafluorophosphate (BOP Reagent)

Bertrand Castro, Geneviève Evin, Claude Selve, +1

Synthesis

EngineeringAmino AcidsBiochemistryPeptide EngineeringBop Reagent +7

Inhibition of human renin by synthetic peptides derived from its prosegment.

Frédéric Cumin, Geneviève Evin, Jean‐Alain Fehrentz, +4

Journal of Biological Chemistry

Molecular PharmacologyMedicinal ChemistryBiochemistryMedicineNatural Sciences +13

Mapping Peptide-binding Domains of the Human V1a Vasopressin Receptor with a Photoactivatable Linear Peptide Antagonist

Sylvie Phalipou, Nathalie de la Cotte, Eric Carnazzi, +5

Journal of Biological Chemistry

Toward Efficient Drug Screening by Homogeneous Assays Based on the Development of New Fluorescent Vasopressin and Oxytocin Receptor Ligands

Laura Albizu, Géraldine Teppaz, René Seyer, +5

Journal of Medicinal Chemistry

Drug TargetPeptide ScienceMolecular PharmacologyNew Fluorescent VasopressinBioanalysis +21

Direct Identification of Human Oxytocin Receptor-binding Domains Using a Photoactivatable Cyclic Peptide Antagonist

Christophe Breton, Hichem Chellil, Majida Kabbaj-Benmansour, +8

Journal of Biological Chemistry

Docking of Linear Peptide Antagonists into the Human V1a Vasopressin Receptor

Sylvie Phalipou, René Seyer, Nathalie de la Cotte, +4

Journal of Biological Chemistry

Peptide ScienceChemical BiologyMedicinal ChemistryBiochemistryPhotochemistry +18

Deglycosylation and fragmentation of purified rat liver angiotensin II receptor: application to the mapping of hormone-binding domains

Franck Désarnaud, Jacky Marie, Colette Lombard, +5

Biochemical Journal

GlycobiologyNew Structural DataChemical BiologyGastrointestinal Peptide HormoneMedicinal Chemistry +18