Pharmacologic Characterization of the Cloned Human Trace Amine-Associated Receptor1 (TAAR1) and Evidence for Species Differences with the Rat TAAR1

David B. Wainscott, Sheila P. Little, Tinggui Yin, +4

Journal of Pharmacology and Experimental Therapeutics

Design of a Potent Combined Pseudopeptide Endothelin-A/Endothelin-B Receptor Antagonist, Ac-<scp>d</scp>Bhg¹⁶-Leu-Asp-Ile-[NMe]Ile-Trp²¹(PD 156252):  Examination of Its Pharmacokinetic and Spectral Properties

Wayne L. Cody, John X. He, Michael D. Reily, +5

Journal of Medicinal Chemistry

Pd 156252Peptide ScienceExperimental PharmacologyGastrointestinal Peptide HormoneMolecular Pharmacology +14

Design of a functional hexapeptide antagonist of endothelin

Wayne L. Cody, Annette M. Doherty, John X. He, +6

Journal of Medicinal Chemistry

Molecular PharmacologyMedicinal ChemistryTranslational PharmacologyNeuropeptidesEndothelinwayne L. Cody +13

Higher Order Structure in the Gas Phase Reflects Solution Structure

Joseph A. Loo, John X. He, Wayne L. Cody

Journal of the American Chemical Society

Crystal StructureEngineeringChemical AnalysisAltmetric Attention ScoreOrganic Chemistry +15

Design and Structure-Activity Relationships of C-Terminal Cyclic Neurotensin Fragment Analogs

Andrea M. Sefler, John X. He, Tomi K. Sawyer, +6

Journal of Medicinal Chemistry

Structure‐activity and conformational studies of a series of modified<i>C</i>‐terminal hexapeptide neurotensin analogues

Deborah Heyl, NDREA M. SEFLER, John X. He, +8

International journal of peptide & protein research

Structure-activity relationships of the potent combined endothelinA/endothelinB receptor antagonist Ac-DDip16-Leu-Asp-Ile-Ile-Trp21 (PD 142893): development of endothelinB receptor selective antagonists

Wayne L. Cody, John X. He, P. L. DePue, +10

Journal of Medicinal Chemistry

Signal TransductionBiochemistryReceptor AffinityMedicineFunctional Selectivity +12

Potent and selective bicyclic lactam inhibitors of thrombin: Part 2: P1 Modifications

Janet S. Plummer, Kent A. Berryman, Cuiman Cai, +15

Bioorganic & Medicinal Chemistry Letters

ThrombosisMedicinal ChemistryPharmaceutical ScienceBiochemistryPart 2 +10

Res-701-1, synthesis and a reevaluation of its effects on the endothelin receptors

John X. He, Wayne L. Cody, Michael A. Flynn, +3

Bioorganic & Medicinal Chemistry Letters

Endothelin ReceptorsMolecular PhysiologySignal TransductionBiochemistryMedicine +5

The design of potent and selective inhibitors of thrombin utilizing a piperazinedione template: Part 1

Wayne L. Cody, Cuiman Cai, Annette M. Doherty, +10

Bioorganic & Medicinal Chemistry Letters

ThrombosisMedicinal ChemistryPart 1BiochemistryPiperazinedione Template +12