John Saunders

Novel 5-HT3 antagonists. Indole oxadiazoles

Christopher J. Swain, Robert J. Baker, Clare O. Kneen et al. · Journal of Medicinal Chemistry · 1991 · 167 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +8

Novel quinuclidine-based ligands for the muscarinic cholinergic receptor

John Saunders, Stephen B. Freedman, Elizabeth A. Harley et al. · Journal of Medicinal Chemistry · 1990 · 158 citations

Medicine, Medicinal Chemistry, Pharmacology +17

Novel benzodiazepine receptor partial agonists: oxadiazolylimidazobenzodiazepines

Frank Wätjen, R. BAKER, Mogens Engelstoff et al. · Journal of Medicinal Chemistry · 1989 · 133 citations

Medicine, Medicinal Chemistry, Pharmacology +6

Synthesis and biological activity of 1,2,4-oxadiazole derivatives: highly potent and efficacious agonists for cortical muscarinic receptors

R. BAKER, T. BOOK, Clare O. Kneen et al. · Journal of Medicinal Chemistry · 1990 · 133 citations

Medicine, Medicinal Chemistry, Pharmacology +17

Discovery of Sodium <i>R</i>-(+)-4-{2-[5-(2-Fluoro-3-methoxyphenyl)-3-(2-fluoro-6-[trifluoromethyl]benzyl)-4-methyl-2,6-dioxo-3,6-dihydro-2<i>H</i>-pyrimidin-1-yl]-1-phenylethylamino}butyrate (Elagolix), a Potent and Orally Available Nonpeptide Antagonist of the Human Gonadotropin-Releasing Hormone Receptor

Chen Chen, Dongpei Wu, Zhiqiang Guo et al. · Journal of Medicinal Chemistry · 2008 · 119 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +16