Kilian Kuhn

Mimicking of Arginine by Functionalized<i>N</i>^ω-Carbamoylated Arginine As a New Broadly Applicable Approach to Labeled Bioactive Peptides: High Affinity Angiotensin, Neuropeptide Y, Neuropeptide FF, and Neurotensin Receptor Ligands As Examples

Max Keller, Kilian Kuhn, Jürgen Einsiedel et al. · Journal of Medicinal Chemistry · 2016 · 41 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +17

High Affinity Agonists of the Neuropeptide Y (NPY) Y₄ Receptor Derived from the C-Terminal Pentapeptide of Human Pancreatic Polypeptide (hPP): Synthesis, Stereochemical Discrimination, and Radiolabeling

Kilian Kuhn, Thomas Ertl, Stefanie Dukorn et al. · Journal of Medicinal Chemistry · 2016 · 26 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +17

N^ω-Carbamoylation of the Argininamide Moiety: An Avenue to Insurmountable NPY Y₁ Receptor Antagonists and a Radiolabeled Selective High-Affinity Molecular Tool ([³H]UR-MK299) with Extended Residence Time

Max Keller, Christoph Hutzler, Kilian Kuhn et al. · Journal of Medicinal Chemistry · 2015 · 25 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +15

Fluorescence- and Radiolabeling of [Lys⁴,Nle^17,30]hPP Yields Molecular Tools for the NPY Y₄Receptor

Stefanie Dukorn, Timo Littmann, Max Keller et al. · Bioconjugate Chemistry · 2017 · 13 citations

Medicine, Biochemistry, Pharmacology +16

In Search of NPY Y₄R Antagonists: Incorporation of Carbamoylated Arginine, Aza-Amino Acids, or<scp>d</scp>-Amino Acids into Oligopeptides Derived from the C-Termini of the Endogenous Agonists

Kilian Kuhn, Timo Littmann, Stefanie Dukorn et al. · ACS Omega · 2017 · 11 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +17