Darius Robinson

Formal total synthesis of FK506. Concise construction of the C(10)-C(34) segment via an effective coupling tactic

Amos B. Smith, Kwunmin Chen, Darius Robinson et al. · Tetrahedron Letters · 1994 · 35 citations

Combinatorial Chemistry, Cross-coupling Reaction, Natural Sciences +6

Discovery, SAR and X-ray structure of 1H-benzimidazole-5-carboxylic acid cyclohexyl-methyl-amides as inhibitors of inducible T-cell kinase (Itk)

K.J.M. Moriarty, Hidenori Takahashi, Steven S. Pullen et al. · Bioorganic & Medicinal Chemistry Letters · 2008 · 32 citations · Full text

Medicinal Chemistry, Drug Target, Biochemistry +12

Itk kinase inhibitors: Initial efforts to improve the metabolical stability and the cell activity of the benzimidazole lead

K.J.M. Moriarty, Michael P. Winters, Lei Qiao et al. · Bioorganic & Medicinal Chemistry Letters · 2008 · 26 citations · Full text

Medicinal Chemistry, Bioorganic Chemistry, Biochemistry +12

5-Aminomethyl-1H-benzimidazoles as orally active inhibitors of inducible T-cell kinase (Itk)

Michael P. Winters, Darius Robinson, Hnin Hnin Khine et al. · Bioorganic & Medicinal Chemistry Letters · 2008 · 24 citations · Full text

Drug Target, Medicine, Drug Discovery +8