Bernd Kaiser

Discovery of 2-Hydroxy-<i>N</i>,<i>N</i>-dimethyl-3-{2-[[(<i>R</i>)-1-(5- methylfuran-2-yl)propyl]amino]-3,4-dioxocyclobut-1-enylamino}benzamide (SCH 527123):  A Potent, Orally Bioavailable CXCR2/CXCR1 Receptor Antagonist

Michael P. Dwyer, Younong Yu, Jianping Chao et al. · Journal of Medicinal Chemistry · 2006 · 116 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +12

Preparation and Detection of Enantiomerically Enriched and Configurationally Stable α‐Thioalkyllithium Compounds

Bernd Kaiser, Dieter Hoppe · Angewandte Chemie International Edition in English · 1995 · 71 citations

Natural Sciences, Chemistry, Organic Chemistry +7

The Configurational Stability of an Enantioenrichedα-Thiobenzyllithium Derivative and the Stereochemical Course of Its Electrophilic Substitution Reactions; Synthesis of Enantiomerically Pure, Tertiary Benzylic Thiols[1,2]

O. Stratmann, Bernd Kaiser, Roland Fröhlich et al. · Chemistry - A European Journal · 2001 · 55 citations

Natural Sciences, Chemistry, Organic Chemistry +10

A Highly Enantiomerically Enriched α‐Thiobenzyl Derivative with Unusual Configurational Stability

Dieter Hoppe, Bernd Kaiser, O. Stratmann et al. · Angewandte Chemie International Edition in English · 1997 · 49 citations

Natural Sciences, Chemistry, Medicinal Chemistry +5

Synthesis and structure–activity relationships of 3,4-diaminocyclobut-3-ene-1,2-dione CXCR2 antagonists

J. Robert Merritt, Laura L. Rokosz, Kingsley H. Nelson et al. · Bioorganic & Medicinal Chemistry Letters · 2006 · 47 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +10